Androgen receptor RTDTs
- Target androgen receptor [AR] and co-target DNA
- Therapeutic uses
- aggressive AR-expressing tumors with high proliferation fraction including virtually all castrate resistant prostate cancers, refractory and recurrent ovarian cancers, and approximately 40% of triple-negative breast cancers
- as an adjuvant to conventional therapy of AR-expressing tumors to kill cancer cells during the DNA repair process
BChE RTDTs
- Target BChE and co-target DNA
- Therapeutic uses
- ovarian cancer
- high risk neuroblastoma with amplified N-MYC
- glioblastoma
- colorectal cancer, particularly hepatic metastases